DDrare
Disease
Drug
Target Gene/Pathway
Contact
JA
Drug
Description in Trials
/
DrugBank
/
KEGG DRUG
Search
A
B
C
D
E
F
G
H
I
J
K
L
M
N
O
P
Q
R
S
T
U
V
W
X
Y
Z
Other
Search results
10
50
100
ALL
descriptions per page:
Showing 1 to 10 of 24 descriptions
Filter by
Reset
|
No.
Drug (Description in trials)
DrugBank
KEGG DRUG
KEGG GENES
KEGG PATHWAY
Disease ID
1
Bosentan
(
Tracleer
(TN))
[1]
Bosentan
Bosentan
(
Tracleer
)
[2]
Bosentan
Bosentan
(
Tracleer
(TN))
,
Bosentan
💬
1. Bosentan
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
1. Bosentan
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[10]
41
41
,
47
,
51
,
84
,
85
,
86
,
88
,
210
,
211
,
212
💬
1. Bosentan
×
Disease ID
Name
41
Giant cell arteritis
47
Buerger disease
51
Scleroderma
84
Sarcoidosis
85
Idiopathic interstitial pneumonia
86
Pulmonary arterial hypertension
88
Chronic thromboembolic pulmonary hypertension
210
Single Ventricle
211
Hypoplastic left heart syndrome
212
Tricuspid atresia
2
Bosentan (
Tracleer
)
[1]
Bosentan
Bosentan
(
Tracleer
)
[2]
Bosentan
Bosentan
(
Tracleer
(TN))
,
Bosentan
💬
2. Bosentan (
Tracleer
)
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
2. Bosentan (
Tracleer
)
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[1]
51
51
💬
2. Bosentan (
Tracleer
)
×
Disease ID
Name
51
Scleroderma
3
Bosentan 125 mg
(
Tracleer
(TN))
[1]
Bosentan
Bosentan
(
Tracleer
)
[2]
Bosentan
Bosentan
(
Tracleer
(TN))
,
Bosentan
💬
3. Bosentan 125 mg
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
3. Bosentan 125 mg
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[1]
51
51
💬
3. Bosentan 125 mg
×
Disease ID
Name
51
Scleroderma
4
Bosentan 62.5 mg
(
Tracleer
(TN))
[1]
Bosentan
Bosentan
(
Tracleer
)
[2]
Bosentan
Bosentan
(
Tracleer
(TN))
,
Bosentan
💬
4. Bosentan 62.5 mg
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
4. Bosentan 62.5 mg
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[1]
51
51
💬
4. Bosentan 62.5 mg
×
Disease ID
Name
51
Scleroderma
5
Bosentan administration
(
Tracleer
(TN))
[1]
Bosentan
Bosentan
(
Tracleer
)
[2]
Bosentan
Bosentan
(
Tracleer
(TN))
,
Bosentan
💬
5. Bosentan administration
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
5. Bosentan administration
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[1]
86
86
💬
5. Bosentan administration
×
Disease ID
Name
86
Pulmonary arterial hypertension
6
Bosentan and Sildenafil
(
Tracleer
(TN))
[2]
Bosentan
Bosentan
(
Tracleer
),
Sildenafil
[3]
Bosentan
Bosentan
(
Tracleer
(TN))
,
Bosentan
,
Sildenafil
💬
6. Bosentan and Sildenafil
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
Sildenafil
Sildenafil (INN)
Aphrodil (TN)
[3]
EDNRA
EDNRA
,
EDNRB
,
PDE5A
💬
6. Bosentan and Sildenafil
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
PDE5A
phosphodiesterase 5A
[11]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Metabolic pathways
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Purine metabolism
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[11]
Calcium signaling pathway
,
Melanogenesis
,
Metabolic pathways
,
Neuroactive ligand-receptor inter
...
[1]
86
86
💬
6. Bosentan and Sildenafil
×
Disease ID
Name
86
Pulmonary arterial hypertension
7
Bosentan group
(
Tracleer
(TN))
[1]
Bosentan
Bosentan
(
Tracleer
)
[2]
Bosentan
Bosentan
(
Tracleer
(TN))
,
Bosentan
💬
7. Bosentan group
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
7. Bosentan group
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[1]
51
51
💬
7. Bosentan group
×
Disease ID
Name
51
Scleroderma
8
BOSENTAN MONOHIDRATO
(
Tracleer
(TN))
[1]
Bosentan
Bosentan
(
Tracleer
)
[2]
Bosentan
Bosentan
(
Tracleer
(TN))
,
Bosentan
💬
8. BOSENTAN MONOHIDRATO
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
8. BOSENTAN MONOHIDRATO
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[1]
86
86
💬
8. BOSENTAN MONOHIDRATO
×
Disease ID
Name
86
Pulmonary arterial hypertension
9
Bosentan monohydrat
(
Tracleer
(TN))
[1]
Bosentan
Bosentan
(
Tracleer
)
[2]
Bosentan
Bosentan
(
Tracleer
(TN))
,
Bosentan
💬
9. Bosentan monohydrat
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
9. Bosentan monohydrat
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[1]
86
86
💬
9. Bosentan monohydrat
×
Disease ID
Name
86
Pulmonary arterial hypertension
10
BOSENTAN MONOHYDRATE
(
Tracleer
(TN))
[1]
Bosentan
Bosentan
(
Tracleer
)
[2]
Bosentan
Bosentan
(
Tracleer
(TN))
,
Bosentan
💬
10. BOSENTAN MONOHYDRATE
×
Name
Other Names
Bosentan
Bosentan (USAN)
Bosentan hydrate (JAN)
Tracleer (TN)
Bosentan
Bosentan (INN)
[2]
EDNRA
EDNRA
,
EDNRB
💬
10. BOSENTAN MONOHYDRATE
×
Name
Full Name
EDNRA
endothelin receptor type A
EDNRB
endothelin receptor type B
[9]
Calcium signaling pathway
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in cancer
,
Relaxin signaling pathway
,
Renin secretion
,
Vascular smooth muscle contraction
,
cAMP signaling pathway
,
cGMP-PKG signaling pathway
💬
[9]
Calcium signaling pathway
,
Melanogenesis
,
Neuroactive ligand-receptor interaction
,
Pathways in c
...
[4]
51
51
,
84
,
86
,
88
💬
10. BOSENTAN MONOHYDRATE
×
Disease ID
Name
51
Scleroderma
84
Sarcoidosis
86
Pulmonary arterial hypertension
88
Chronic thromboembolic pulmonary hypertension